Identifiers | ||
Product Name | Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016) | |
Catalogue No. | CM726481 | |
Description | Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer models. | |
Application | 100 mg. Purity >99%. CAS# 388082-78-8. Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer model | |
CAS Number | 388082-78-8 | |
Formula | C₂₉H₂₆ClFN₄O₄S.2C₇H₈O₃S | |
MW | 925.46 | |
Storage Condition | -20°C |
Brand | Packing | Pricing | Quote request |
IL | 100 mg | Inquiry | Ask Quote |
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